Synthesis, Characterization and in Vitro Evaluation of MRSA Inhibitors by Designing of Ligand Based Approach (QSAR)

Authors

  • Nilesh S. Pawar  Synthetic Research Laboratory Department of Chemistry Pratap College, Amalner, Maharashtra, India
  • Milind S. Thakare  Applied Science Department, R. C. Patel Institute of Technology, Shirpur, Maharashtra, India
  • Pramod N. Patil  

Keywords:

QSAR, Thiabendazole derivative, MRSA, Pharmacological activities.

Abstract

In present investigation, we have design, synthesize and evaluate methicillin-resistant staphylococcus aureus (MRSA) inhibitors. It appears interesting result of MRSA inhibitors. Newly synthesized compounds have been characterized and studied their antimicrobial activity especially MRSA gram positive bacterium. The compounds were found to exhibit good to comparable activity with respect to standards.

References

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International Journal of Scientific Research in Science, Engineering and Technology

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Published

2018-02-28

Issue

Volume 4, Issue 1, January-February-2018

Section

Research Articles

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This work is licensed under a Creative Commons Attribution 4.0 International License.

How to Cite

[1]
Nilesh S. Pawar, Milind S. Thakare, Pramod N. Patil, " Synthesis, Characterization and in Vitro Evaluation of MRSA Inhibitors by Designing of Ligand Based Approach (QSAR), International Journal of Scientific Research in Science, Engineering and Technology(IJSRSET), Print ISSN : 2395-1990, Online ISSN : 2394-4099, Volume 4, Issue 1, pp.908-912, January-February-2018.