Synthesis and Biological Evaluation of Some New Acetyl Pyrazoline Derivatives of 3-Aryl-2-Isobutanoyl-N-Phenyl-Acrylamide

Authors(1) :-D. N. Joshi

The broad spectrums of pharmacological properties have been demonstrated by the pyrazole nucleus. Some new 1-Acetyl-5-aryl-3-isopropyl-4-[n-phenyl-aminocarbonyl]-4,5-dihydro-1H-pyrazoles.The pyrazoline derivatives of Type (1a-j) have been synthesized by the reaction of 3-Aryl-2-isobutanoyl-N-phenyl-acrylamide with hydrazine hydrate in glacial acetic acid. All the prepared compounds were characterized by their spectral (I.R., N.M.R., Mass) data and screened for their antimicrobial activities.

Authors and Affiliations

D. N. Joshi
Department of Chemistry, R.R.Mehta College of Science & C.L.Parikh college of Commerce Palanpur, Gujarat, India

3-Aryl-2-isobutanoyl-N-phenyl-acrylamide, Acetyl pyrazoles, Antimicrobial activities.

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Publication Details

Published in : Volume 1 | Issue 1 | 2014
Date of Publication : 2014-12-30
License:  This work is licensed under a Creative Commons Attribution 4.0 International License.
Page(s) : 169-173
Manuscript Number : IJSRSET1849118
Publisher : Technoscience Academy

Print ISSN : 2395-1990, Online ISSN : 2394-4099

Cite This Article :

D. N. Joshi, " Synthesis and Biological Evaluation of Some New Acetyl Pyrazoline Derivatives of 3-Aryl-2-Isobutanoyl-N-Phenyl-Acrylamide, International Journal of Scientific Research in Science, Engineering and Technology(IJSRSET), Print ISSN : 2395-1990, Online ISSN : 2394-4099, Volume 1, Issue 1, pp.169-173, .2014
URL : http://ijsrset.com/IJSRSET1849118

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